PROTAC ERRα ligand 2
CAS No. 2306388-57-6
PROTAC ERRα ligand 2 ( —— )
产品货号. M20565 CAS No. 2306388-57-6
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥713 | 有现货 |
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5MG | ¥1191 | 有现货 |
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10MG | ¥1596 | 有现货 |
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25MG | ¥3208 | 有现货 |
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50MG | ¥4836 | 有现货 |
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100MG | ¥6901 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称PROTAC ERRα ligand 2
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
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产品描述PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM).
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同义词——
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通路Endocrinology/Hormones
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靶点Estrogen Receptor/ERR
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受体ERRα
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研究领域——
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适应症——
化学信息
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CAS Number2306388-57-6
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分子量445.31
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分子式C20H13F6NO4
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纯度>98% (HPLC)
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溶解度——
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SMILESCOc1cc(\C=C(/C#N)C(O)=O)ccc1OCc1ccc(cc1C(F)(F)F)C(F)(F)F
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Peng L Zhang Z Lei C et al. Identification of New Small-Molecule Inducers of Estrogen-Related Receptor alpha (ERRa) Degradation[J]. ACS Medicinal Chemistry Letters 2019 10(5).
产品手册
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